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Oral drug solutions

Syrups: contains ↑ sugar concentration.   Sweet and viscous.     Syrup NF (simple syrup): 85% w/v sugar.   Sugars have low...




Syrups: contains ↑ sugar concentration.  Sweet and viscous.   

Syrup NF (simple syrup): 85% w/v sugar.  Sugars have low solvent capacity for water soluble drugs because hydrogen bonding between sugar and water is very strong.  Dilute sucrose solutions are excellent media for microbial growth.  As sugar concentration approaches saturation, the solution becomes self-preserved, however temperature fluctuations may cause sugar crystallization.  Syrup USP  is self-preserved with ↓ crystallization potential.  

Elixirs: contain alcohol as a solvent (5-40%).  Elixirs become turbid when diluted by aqueous liquids.  Alcohol ↑ salt taste.  Salts also have limited solubility in alcohol.   

Aromatic elixir NF: mixture of two alcohol  concentrations resulting in 22% alcohol.  

Aromatic waters:  are saturated aqueous solutions of volatile oils.  Used for flavoring.  Stored in tight, light resistant containers.  Adding large amount of water soluble drug may cause insoluble layer to form (salting out) due to better attraction with the water solvent than the oils.  

Spirits (essences): volatile substances in 50-90% alcohol.  It water is added, oils separate.  Used medicinally or as flavors.  Store in tight containers.  

Tinctures:   stable alcohol solutions of chemicals or soluble constituents or vegetable drugs.  Prepared using extraction using maceration or percolation.  Alcohol content varies widely.  

Fluidextracts:  liquid extracts of vegetable drugs that contain alcohol as a solvent, preservative, or both.   Prepared by percolation.  Ten times as concentrated and potent as tinctures (100% vs. 10%). 

Mouthwashes: use alcohol or glycerin to dissolve volatile ingredients.

Astringents: locally applied solutions that ppt protein.  Astringents ↓ cell permeability without causing injury.  They cause constriction, wrinkling and blanching of skin.  They ↓ secretions and are used as antiperspirants.  Examples: alulminum acetate, aluminum subacetate, calcium hydroxide.
Antibacterial topical solutions:  e.g. benzalkonium chloride, strong iodine, providone-iodine. .

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